其他產品及廠家
(z)-tyrphostin a51 is the z configuration of lanoconazole a51. tyrphostin a51 is a potent protein tyrosine kinase (ptk) inhibitor which inhibits the volume-sensitive release of [3 h]taurine in primary astrocyte cultures in a dose-dependent manner. tyrphostin a51 markedly reduces cellular tyrosyl phosphorylation level. tyrphostin a51 inhibits both basal and egf-induced human bone cell proliferation [1] [2].
更新時間:2025-12-04
tyrphostin ag957, a tyrosine kinase inhibitor with anti-bcr/abl tyrosine kinase activity restores beta1 integrin-mediated adhesion and inhibitory signaling in chronic myelogenous leukemia hematopoietic progenitors[1].
更新時間:2025-12-04
apogossypolone (apog2) is a semi-synthesized derivative of gossypol which is a nonpeptidic small molecule inhibitor targeting bcl-2 family proteins with k i values of 35, 25 and 660 nm for bcl-2, mcl-1 and bcl-x l, respectively. apogossypolone shows antitumor activities, induces cell apoptosis [1] and autophagy [2]. apogossypolone also has antifungal activity [3].
更新時間:2025-12-04
azepexole dihydrochloride (b-ht 933), a potent and selective alpha 2-adrenoceptor agonist, exhibits affinity for α2a-, α2b-, and α2c-adrenoceptor subtypes with pkis of 8.3, 7.6, and 7.5, respectively [1]. it elicits a concentration-dependent inhibition of peristaltic contractions, evidenced by an ic50 of 78.72 nm.
更新時間:2025-12-04
azepexole hydrochloride (4h-oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-adrenoceptor agonist with anaesthetic effects.
更新時間:2025-12-04
bd 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (ki = 2 nm). bd 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors.
更新時間:2025-12-04
triptolide (pg490) belongs to the tricyclic diterpenoid group of natural products and is an inhibitor of nf-κb activation. triptolide exhibits immunosuppressive, anti-rheumatic, anti-inflammatory, anti-proliferative and anti-tumor activities.
更新時間:2025-12-04
bms 182874 hydrochloride is a nonpeptide endothelin (el) receptor antagonist.
更新時間:2025-12-04
cgp 3466b maleate (omigapil maleate) is an orally bioavailable gapdh nitrosylation inhibitor. omigapil maleate abrogates aβ1-42-induced tau acetylation, memory impairment, and locomotor dysfunction in mice. omigapil maleate has the potential for the research of alzheimer´s disease. omigapil maleate (cgp3446b maleate) is a apoptosis inhibitor. omigapil maleate can be used for the research of congenital muscular dystrophy (cmd).
更新時間:2025-12-04
crt5, a pyrazine benzamide, is a potent and selective pkd inhibitor. the vegf-induced phosphorylation of three pkd substrates (ic50s = 1, 2, and 1.5 nm for pkd1, pkd2, and pkd3, respectively), histone deacetylase 5, creb (camp-response-element-binding protein), and hsp27 (heat-shock protein 27) at ser82, is also inhibited by crt5. crt5 decreases vegf-induced endothelial migration, proliferation, and tubulogenesis[1].
更新時間:2025-12-04
dynamin inhibitory peptide acetate is a peptide with the sequence gln-val-pro-ser-arg-pro-asn-arg-ala-pro that inhibit the gtpase dynamin.
更新時間:2025-12-04
hexythiazox is a mite growth regulator and a thiazolidine based acaricide that has long-lasting effects against many kinds of mites and is applied at any stage of the plant growth from budding to fruiting.
更新時間:2025-12-04
guanylyl imidodiphosphate trisodium (guanosine 5´-[β,γ-imido]triphosphate), a non-hydrolysable gtp analogue, activates adp-ribosylation factor (arf) and strongly stimulates adenylate cyclase. it is utilized in protein synthesis studies [1] [2] [3].
更新時間:2025-12-04
gw 610 is an antitumor benzothiazole that shows growth-inhibitory activity against several cancer cell lines. in mcf-7 and mda 468 human cancer cell lines, potent antiproliferative activity (growth inhibition (gi50) < 0.1 nm) was observed.
更新時間:2025-12-04
inca-6 (triptycene-1,4-quinone) is a cell-permeable nfat inhibitor. inca-6 inhibits of cn-nfat signaling by targeting of nfat(p) substrate to the calcineurin (cn) phosphatase site.
更新時間:2025-12-04
inotilone is a major component of inonotus linteus, a traditional chinese medical herb and can be used for research of metastatic lung cancer cells.
更新時間:2025-12-04
lh-21 is a potent in vivo neutral cannabinoid cb1 receptor antagonist. lh-21 reduces food intake and body weight gain in obese zucker rats., and results in a dose-dependent inhibition of feeding [1].
更新時間:2025-12-04
lt175, a dual pparα/γ ligand, demonstrates potent insulin-sensitizing effects while exhibiting reduced adipogenic properties. this compound is an orally active partial agonist targeting pparγ, with ec50 values of 0.22 μm for hpparα, 0.26 μm for mpparα, and 0.48 μm for hpparγ. lt175 specifically interacts with pparγ, influencing the recruitment of coregulators such as the cyclic-amp response element-binding protein-binding protein and nuclear corepressor 1 (ncor1). additionally, lt175´s int
更新時間:2025-12-04
oac3 (4-fluoro-n-(1h-indol-5-yl)benzamide) is an activator of octamer-bound transcription factor 4.
更新時間:2025-12-04
ono-4817 is a broad-spectrum matrix metalloproteinase (mmp) inhibitor that potentially mitigates atherosclerotic neointimal proliferation and atheromatous plaque progression by suppressing matrix metalloproteinases (mmps). it effectively reduces the development of aortic intimal hyperplasia in experimental hyperlipidemic rabbits [1].
更新時間:2025-12-04
ono-rs-082 is a ca2+-independent phospholipase a2 inhibitor.?
更新時間:2025-12-04
oxa-01 is a potent mtorc1 and mtorc2 inhibitor, with ic 50 values of 29 nm and 7 nm, respectively [1]. oxa-01 demonstrates broad anti-tumor activity.
更新時間:2025-12-04
pregnenolone carbonitrile (5-pregnen-3β-ol-20-one-16α-carbonitrile) is an activator of rodent-pxr and induces the expression of cyp3a.
更新時間:2025-12-04
psora-4 is a potent and selective inhibitor of k v 1.3 (voltage-gated potassium channels) with a hill coefficient of 2 and an ec50 value of 3 nm [1]. psora-4 has immunosuppressive activity and inhibits proliferation of human and rat myelin-specific effector memory t cells in vitro [2].
更新時間:2025-12-04
resistomycin (geliomycin), a pentacyclic polyketide antibiotic, exhibits potent anticancer properties by triggering apoptosis.
更新時間:2025-12-04
rev 5901 is a competitive and orally effective antagonist of leukotriene receptor, with a ki of 0.7 μm. rev 5901 is also a 5-lipoxygenase inhibitor. rev 5901 can be used for the research of asthma in which leukotriene release be involved [1] [2].
更新時間:2025-12-04
rev 5901a (rev 5901 hcl) is an orally active leukotriene receptor antagonist and 5-lipoxygenase inhibitor with antimicrobial activity that attenuates colon cancer growth in mice.rev 5901a has been used in studies of asthma and myocardial infarction. rev 5901a is used to study asthma and myocardial infarction.
更新時間:2025-12-04
sephin1 (ifb-088) is reportedly a selective inhibitor of gadd34 (ppp1r15a), which is a stress-induced regulatory subunit of protein phosphatase 1 complex that dephosphorylates eif2α
更新時間:2025-12-04
tae-1 is an inhibitor of amyloid-β fibril formation and aggregation. it inhibits cholinesterases ache and buche with ic50 of 0.3 μm and 3.9 μm, respectively.
更新時間:2025-12-04
tc-e 5003 (nsc-30176) is a selective inhibitor of prmt1 with ic50 of 1.5 μm.
更新時間:2025-12-04
ucm05 (g28ucm) is a potent inhibitor of fatty acid synthase (fasn) with efficacy against her2+ breast cancer xenografts, including in cell lines resistant to anti-her2 drugs [1]. additionally, it functions as an inhibitor of the filamentous temperature-sensitive protein z (ftsz), selectively inhibiting the growth of the gram-positive bacterium b. subtilis with minimum inhibitory concentration (mic) values of 100 μm, while showing no activity against the gram-negative bacterium e. coli [2].
更新時間:2025-12-04
sepantronium hydrochloride (ym-155 hydrochloride) is a novel survivin suppressant that inhibits survivin promoter with an ic 50 of 0.54 nm[1].
更新時間:2025-12-04
z-lehd-fmk is a selective and potent caspase-9 inhibitor that protects against reperfusion injury and slows apoptosis.z-lehd-fmk exhibits antitumor and neuroprotective activity, increases the yield of in vitro-produced preimplantation embryos of bubalus bubalis and alters the cellular stress response.
更新時間:2025-12-04
zileuton sodium (a 64077 sodium) is a potent and selective inhibitor of 5-lipoxygenase with anti-inflammatory activities.
更新時間:2025-12-04
1-naphthyl 3,5-dinitrobenzoate (jmc-4) is an inhibitor of 5-lox can be used in studies about inflammatory therapy.
更新時間:2025-12-04
sulfachloropyridazine (sulfachlorpyridazine) is a sulfonamide antimicrobial used for urinary tract infections and in veterinary medicine.
更新時間:2025-12-04
(±)-hexanoylcarnitine chloride is a fatty acid metabolite that breaks down fatty acids into small compounds that can be utilized by the body. (±)-hexanoylcarnitine chloride can be used as a biomarker by being specific for rat skeletal muscle toxicity.
更新時間:2025-12-04
2-fluoropalmitic acid, functioning as an acyl-coa synthetase inhibitor, is a potential anti-glioma agent. it diminishes the viability and stem-like characteristics of glioma stem cells (gscs) and hinders the proliferation and invasion of glioma cell lines [1].
更新時間:2025-12-04
gemsa is a potent inhibitor of enkephalin convertase ( k i =8.8 nm) with analgesic effect[1].
更新時間:2025-12-04
a-841720 is a potent, selective, and non-competitive antagonist of the mglu1 receptor, exhibiting an ic 50 value of 10 nm specifically for the human mglu1 receptor. it demonstrates a 34-fold greater selectivity for mglu1 over mglu5 (ic 50 of 342 nm), with negligible activity across a spectrum of other neurotransmitter receptors, ion channels, and transporters. additionally, a-841720 possesses analgesic potential within a certain dose range [1] [2].
更新時間:2025-12-04
sulfamethazine sodium (sulfadimethyldiazine sodium salt) salt is a sodium salt form of sulfamethazine, a sulfonamide antibiotic used in the livestock industry.
更新時間:2025-12-04
l-ascorbic acid 2-phosphate trisodium (sodium ascorbyl phosphate) is used in biocatalytic dephosphorylation for electric power generation and electrochemical detection assays.
更新時間:2025-12-04
act-335827 is an orally available, brain-penetrant orexin type 1 receptor selective antagonist. act-33582 acts on oxr1 and oxr2 with ic 50 values of 6 nm and 417 nm, respectively. act-33582 can be used in studies related to neurological disorders [1].
更新時間:2025-12-04
aeg 3482 is a potent antiapoptotic compound. aeg 3482 inhibits jun kinase (jnk) activity through induced expression of heat shock protein 70 (hsp70). aeg 3482 directly binds hsp90, thereby facilitating hsf1-dependent expression of hsp70 and hsp25.
更新時間:2025-12-04
ag 556 is a selective inhibitor of egfr and blocks lps-induced tnf-α production.
更新時間:2025-12-04
arm1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. the ic50 values are 7.61 ?m for aminopeptidase and 12.4 ?m for epoxide hydrolase.
更新時間:2025-12-04
tris(2,2,2-trifluoroethyl) borate (sl 75212) is mostly used in condensation reactions. it has been shown to promote the direct formation of amides from carboxylic acids and amines as well as the formation of imines from amines or amides with carbonyl compounds.
更新時間:2025-12-04
asterric acid is a useful organic compound for research related to life sciences. the catalog number is t21860 and the cas number is 577-64-0.
更新時間:2025-12-04
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