其他產(chǎn)品及廠家

VU0359595；化合物VU0359595VU0359595-1|||CID-53361951|||ML-270；VU0359595-1|||CID-53361951|||ML-270
vu0359595 (ml-270) is a potent and selective pharmacological phospholipase d1 (pld1) inhibitor with an ic50 of 3.7 nm. vu0359595 is >1700-fold selective for pld1 over pld2 (ic50 of 6.4 μm). vu0359595 can be used for the research of cancer, diabetes, neurodegenerative and inflammatory diseases.
更新時間:2025-12-04
10-DEBC hydrochloride；化合物 T2177810-DEBC hydrochloride
10-debc hydrochloride, a selective akt inhibitor demonstrating an ic50 value of 1.28 μm, is identified as a novel anti-tuberculosis compound [1] [2].
更新時間:2025-12-04
AMI5；化合物AMI-5AMI 5|||Eosin Y Disodium|||AMI-5；AMI 5|||Eosin Y Disodium|||AMI-5
ami5 (eosin y disodium) is a versatile red dye used in cosmetics, pharmaceuticals, textiles, etc., and as tissue stain, vital stain, and counterstain with hematoxylin. it is also used in special culture media.
更新時間:2025-12-04
A-286982；化合物A 286982A-286982
a 286982 is an inhibitor that blocks the integrin-ligand interaction between leukocyte function-associated antigen-1 (lfa-1) and intercellular adhesion molecule-1.
更新時間:2025-12-04
A 77636 hydrochloride；鹽酸A77636A77636 hydrochloride；鹽酸A77636|||A77636 hydrochloride
a 77636 hydrochloride is a potent, orally active, selective and long acting dopamine d1 receptor agonist (pki=7.40; ki=39.8 nm). a 77636 hydrochloride shows antiparkinsonian activity. a 77636 hydrochloride is functionally inactive at dopamine d2 receptor.
更新時間:2025-12-04
AG-183；化合物 T21783AG-183
(z)-tyrphostin a51 is the z configuration of lanoconazole a51. tyrphostin a51 is a potent protein tyrosine kinase (ptk) inhibitor which inhibits the volume-sensitive release of [3 h]taurine in primary astrocyte cultures in a dose-dependent manner. tyrphostin a51 markedly reduces cellular tyrosyl phosphorylation level. tyrphostin a51 inhibits both basal and egf-induced human bone cell proliferation [1] [2].
更新時間:2025-12-04
AG957；化合物Tyrphostin AG957u00A0AG957
tyrphostin ag957, a tyrosine kinase inhibitor with anti-bcr/abl tyrosine kinase activity restores beta1 integrin-mediated adhesion and inhibitory signaling in chronic myelogenous leukemia hematopoietic progenitors[1].
更新時間:2025-12-04
Apogossypolone (ApoG2)；化合物 T21786Apogossypolone (ApoG2)
apogossypolone (apog2) is a semi-synthesized derivative of gossypol which is a nonpeptidic small molecule inhibitor targeting bcl-2 family proteins with k i values of 35, 25 and 660 nm for bcl-2, mcl-1 and bcl-x l, respectively. apogossypolone shows antitumor activities, induces cell apoptosis [1] and autophagy [2]. apogossypolone also has antifungal activity [3].
更新時間:2025-12-04
B-HT 933 dihydrochloride；化合物 T21787B-HT 933 dihydrochloride
azepexole dihydrochloride (b-ht 933), a potent and selective alpha 2-adrenoceptor agonist, exhibits affinity for α2a-, α2b-, and α2c-adrenoceptor subtypes with pkis of 8.3, 7.6, and 7.5, respectively [1]. it elicits a concentration-dependent inhibition of peristaltic contractions, evidenced by an ic50 of 78.72 nm.
更新時間:2025-12-04
Azepexole hydrochloride；化合物T21787L4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydr
azepexole hydrochloride (4h-oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-adrenoceptor agonist with anaesthetic effects.
更新時間:2025-12-04
BD 1008 dihydrobromide；N-[2-(3,4-二氯苯基)乙基]-N-甲基-1-吡咯烷乙胺二氫溴酸鹽BD 1008 dihydrobromide
bd 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (ki = 2 nm). bd 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors.
更新時間:2025-12-04
Triptolide；雷公藤甲素PG490|||NSC 163062；PG490|||NSC 163062|||雷公藤甲素
triptolide (pg490) belongs to the tricyclic diterpenoid group of natural products and is an inhibitor of nf-κb activation. triptolide exhibits immunosuppressive, anti-rheumatic, anti-inflammatory, anti-proliferative and anti-tumor activities.
更新時間:2025-12-04
BMS 182874 hydrochloride；化合物BMS 182874 hydrochlorideBMS 182874 hydrochloride
bms 182874 hydrochloride is a nonpeptide endothelin (el) receptor antagonist.
更新時間:2025-12-04
CGP 3466B maleate馬來酸CGP3466B馬來酸CGP3466B|||Omigapil (Maleate)|||Omigapil maleate
cgp 3466b maleate (omigapil maleate) is an orally bioavailable gapdh nitrosylation inhibitor. omigapil maleate abrogates aβ1-42-induced tau acetylation, memory impairment, and locomotor dysfunction in mice. omigapil maleate has the potential for the research of alzheimer´s disease. omigapil maleate (cgp3446b maleate) is a apoptosis inhibitor. omigapil maleate can be used for the research of congenital muscular dystrophy (cmd).
更新時間:2025-12-04
CRT5；化合物 T21795CRT5
crt5, a pyrazine benzamide, is a potent and selective pkd inhibitor. the vegf-induced phosphorylation of three pkd substrates (ic50s = 1, 2, and 1.5 nm for pkd1, pkd2, and pkd3, respectively), histone deacetylase 5, creb (camp-response-element-binding protein), and hsp27 (heat-shock protein 27) at ser82, is also inhibited by crt5. crt5 decreases vegf-induced endothelial migration, proliferation, and tubulogenesis[1].
更新時間:2025-12-04
Dynamin inhibitory peptide Acetate；化合物T21798LDynamin inhibitory peptide Acetate(251634-21-6 Free bas
dynamin inhibitory peptide acetate is a peptide with the sequence gln-val-pro-ser-arg-pro-asn-arg-ala-pro that inhibit the gtpase dynamin.
更新時間:2025-12-04
Hexythiazox；噻螨酮Hexythiazox
hexythiazox is a mite growth regulator and a thiazolidine based acaricide that has long-lasting effects against many kinds of mites and is applied at any stage of the plant growth from budding to fruiting.
更新時間:2025-12-04
Guanylyl Imidodiphosphate；化合物 T21803Guanylyl Imidodiphosphate
guanylyl imidodiphosphate trisodium (guanosine 5´-[β,γ-imido]triphosphate), a non-hydrolysable gtp analogue, activates adp-ribosylation factor (arf) and strongly stimulates adenylate cyclase. it is utilized in protein synthesis studies [1] [2] [3].
更新時間:2025-12-04
GW 610；化合物GW 610GW 610
gw 610 is an antitumor benzothiazole that shows growth-inhibitory activity against several cancer cell lines. in mcf-7 and mda 468 human cancer cell lines, potent antiproliferative activity (growth inhibition (gi50) < 0.1 nm) was observed.
更新時間:2025-12-04
HNHA；N-羥基-7-(2-萘硫基)-庚酰胺HNHA
hnha is an inhibitor of hdac.
更新時間:2025-12-04
INCA-6化合物INCA-6Triptycene-1,4-quinone
inca-6 (triptycene-1,4-quinone) is a cell-permeable nfat inhibitor. inca-6 inhibits of cn-nfat signaling by targeting of nfat(p) substrate to the calcineurin (cn) phosphatase site.
更新時間:2025-12-04
Inotilone；化合物InotiloneInotilone
inotilone is a major component of inonotus linteus, a traditional chinese medical herb and can be used for research of metastatic lung cancer cells.
更新時間:2025-12-04
LH 21；化合物 T21811LH 21
lh-21 is a potent in vivo neutral cannabinoid cb1 receptor antagonist. lh-21 reduces food intake and body weight gain in obese zucker rats., and results in a dose-dependent inhibition of feeding [1].
更新時間:2025-12-04
LT175；化合物 T21812LT175|||LT 175|||LT-175|||LT175；0
lt175, a dual pparα/γ ligand, demonstrates potent insulin-sensitizing effects while exhibiting reduced adipogenic properties. this compound is an orally active partial agonist targeting pparγ, with ec50 values of 0.22 μm for hpparα, 0.26 μm for mpparα, and 0.48 μm for hpparγ. lt175 specifically interacts with pparγ, influencing the recruitment of coregulators such as the cyclic-amp response element-binding protein-binding protein and nuclear corepressor 1 (ncor1). additionally, lt175´s int
更新時間:2025-12-04
OAC3；化合物OAC34-fluoro-N-(1H-indol-5-yl)benzamide；4-fluoro-N-(1H-indol-5-yl)benzamide
oac3 (4-fluoro-n-(1h-indol-5-yl)benzamide) is an activator of octamer-bound transcription factor 4.
更新時間:2025-12-04
ONO 4817；化合物 T21814ONO 4817
ono-4817 is a broad-spectrum matrix metalloproteinase (mmp) inhibitor that potentially mitigates atherosclerotic neointimal proliferation and atheromatous plaque progression by suppressing matrix metalloproteinases (mmps). it effectively reduces the development of aortic intimal hyperplasia in experimental hyperlipidemic rabbits [1].
更新時間:2025-12-04
ONO-RS-082；化合物ONO-RS-082ONO-RS-082
ono-rs-082 is a ca2+-independent phospholipase a2 inhibitor.?
更新時間:2025-12-04
OXA-01；化合物 T21816OXA-01
oxa-01 is a potent mtorc1 and mtorc2 inhibitor, with ic 50 values of 29 nm and 7 nm, respectively [1]. oxa-01 demonstrates broad anti-tumor activity.
更新時間:2025-12-04
Pregnenolone Carbonitrile化合物Pregnenolone CarbonitrilePregnenolone 16α-carbonitrileu00A0|||5-Pregnen-
pregnenolone carbonitrile (5-pregnen-3β-ol-20-one-16α-carbonitrile) is an activator of rodent-pxr and induces the expression of cyp3a.
更新時間:2025-12-04
Psora 4；化合物 T21819Psora 4
psora-4 is a potent and selective inhibitor of k v 1.3 (voltage-gated potassium channels) with a hill coefficient of 2 and an ec50 value of 3 nm [1]. psora-4 has immunosuppressive activity and inhibits proliferation of human and rat myelin-specific effector memory t cells in vitro [2].
更新時間:2025-12-04
Resistomycin；硫酸卡那霉素Geliomycin|||Heliomycin；Geliomycin|||Heliomycin
resistomycin (geliomycin), a pentacyclic polyketide antibiotic, exhibits potent anticancer properties by triggering apoptosis.
更新時間:2025-12-04
REV 5901；化合物 T21821REV 5901
rev 5901 is a competitive and orally effective antagonist of leukotriene receptor, with a ki of 0.7 μm. rev 5901 is also a 5-lipoxygenase inhibitor. rev 5901 can be used for the research of asthma in which leukotriene release be involved [1] [2].
更新時間:2025-12-04
REV 5901A；化合物 REV 5901AREV 5901 HCl|||REV 5901A（101910-24-1 Free base）；REV 5901 HCl|||REV 5901A（1019
rev 5901a (rev 5901 hcl) is an orally active leukotriene receptor antagonist and 5-lipoxygenase inhibitor with antimicrobial activity that attenuates colon cancer growth in mice.rev 5901a has been used in studies of asthma and myocardial infarction. rev 5901a is used to study asthma and myocardial infarction.
更新時間:2025-12-04
Sephin1；化合物Sephin1NSC 65390|||IFB-088；NSC 65390|||IFB-088
sephin1 (ifb-088) is reportedly a selective inhibitor of gadd34 (ppp1r15a), which is a stress-induced regulatory subunit of protein phosphatase 1 complex that dephosphorylates eif2α
更新時間:2025-12-04
TAE-1；化合物TAE-1TAE-1
tae-1 is an inhibitor of amyloid-β fibril formation and aggregation. it inhibits cholinesterases ache and buche with ic50 of 0.3 μm and 3.9 μm, respectively.
更新時間:2025-12-04
TC-E 5003化合物TC-E 5003NSC 30176
tc-e 5003 (nsc-30176) is a selective inhibitor of prmt1 with ic50 of 1.5 μm.
更新時間:2025-12-04
UCM05；化合物UCM05G28UCM；G28UCM
ucm05 (g28ucm) is a potent inhibitor of fatty acid synthase (fasn) with efficacy against her2+ breast cancer xenografts, including in cell lines resistant to anti-her2 drugs [1]. additionally, it functions as an inhibitor of the filamentous temperature-sensitive protein z (ftsz), selectively inhibiting the growth of the gram-positive bacterium b. subtilis with minimum inhibitory concentration (mic) values of 100 μm, while showing no activity against the gram-negative bacterium e. coli [2].
更新時間:2025-12-04
YM-155 hydrochloride；化合物 T21834YM-155 hydrochloride
sepantronium hydrochloride (ym-155 hydrochloride) is a novel survivin suppressant that inhibits survivin promoter with an ic 50 of 0.54 nm[1].
更新時間:2025-12-04
Z-LEHD-fmk；多肽Z-LEHD-fmkZ-LEHD-fmk
z-lehd-fmk is a selective and potent caspase-9 inhibitor that protects against reperfusion injury and slows apoptosis.z-lehd-fmk exhibits antitumor and neuroprotective activity, increases the yield of in vitro-produced preimplantation embryos of bubalus bubalis and alters the cellular stress response.
更新時間:2025-12-04
Zileuton sodium；化合物 T21836Zileuton sodium
zileuton sodium (a 64077 sodium) is a potent and selective inhibitor of 5-lipoxygenase with anti-inflammatory activities.
更新時間:2025-12-04
1-Naphthyl 3,5-dinitrobenzoate；化合物1-Naphthyl 3,5-dinitrobenzoateJMC-4；JMC-4
1-naphthyl 3,5-dinitrobenzoate (jmc-4) is an inhibitor of 5-lox can be used in studies about inflammatory therapy.
更新時間:2025-12-04
10Panx Acetate；化合物10Panx Acetate10Panx Acetate(955091-53-9 Free base)；10Panx Acetate(955091-53-9 Fre
10panx acetate is a mimetic inhibitory peptide that readily and reversibly inhibits the panx1 currents.
更新時間:2025-12-04
Sulfachloropyridazine磺胺二甲基嘧啶Sulfachlorpyridazine|||磺胺二甲基嘧啶
sulfachloropyridazine (sulfachlorpyridazine) is a sulfonamide antimicrobial used for urinary tract infections and in veterinary medicine.
更新時間:2025-12-04
(±)-Hexanoylcarnitine chloride(±)-氯化己酰肉堿DL-Hexanoylcarnitine chloride
(±)-hexanoylcarnitine chloride is a fatty acid metabolite that breaks down fatty acids into small compounds that can be utilized by the body. (±)-hexanoylcarnitine chloride can be used as a biomarker by being specific for rat skeletal muscle toxicity.
更新時間:2025-12-04
2-fluoro Palmitic Acid；化合物 T218422-fluoro Palmitic Acid
2-fluoropalmitic acid, functioning as an acyl-coa synthetase inhibitor, is a potential anti-glioma agent. it diminishes the viability and stem-like characteristics of glioma stem cells (gscs) and hinders the proliferation and invasion of glioma cell lines [1].
更新時間:2025-12-04
GEMSA；化合物 GEMSAGEMSA
gemsa is a potent inhibitor of enkephalin convertase ( k i =8.8 nm) with analgesic effect[1].
更新時間:2025-12-04
A 841720；化合物 T21848A 841720
a-841720 is a potent, selective, and non-competitive antagonist of the mglu1 receptor, exhibiting an ic 50 value of 10 nm specifically for the human mglu1 receptor. it demonstrates a 34-fold greater selectivity for mglu1 over mglu5 (ic 50 of 342 nm), with negligible activity across a spectrum of other neurotransmitter receptors, ion channels, and transporters. additionally, a-841720 possesses analgesic potential within a certain dose range [1] [2].
更新時間:2025-12-04
Sulfamethazine sodium；磺胺二甲嘧啶鈉Sulfadimethyldiazine Sodium Salt|||Sulfamethazine sodium salt；Sulfadime
sulfamethazine sodium (sulfadimethyldiazine sodium salt) salt is a sodium salt form of sulfamethazine, a sulfonamide antibiotic used in the livestock industry.
更新時間:2025-12-04
L-Ascorbic acid 2-phosphate trisodium；L-抗壞血酸-2-磷酸三鈉鹽L-Ascorbic acid 2-phosphate trisodium salt|||Sod
l-ascorbic acid 2-phosphate trisodium (sodium ascorbyl phosphate) is used in biocatalytic dephosphorylation for electric power generation and electrochemical detection assays.
更新時間:2025-12-04
ACT 335827；化合物 T21850ACT 335827
act-335827 is an orally available, brain-penetrant orexin type 1 receptor selective antagonist. act-33582 acts on oxr1 and oxr2 with ic 50 values of 6 nm and 417 nm, respectively. act-33582 can be used in studies related to neurological disorders [1].
更新時間:2025-12-04

最新產(chǎn)品

熱門儀器： 液相色譜儀 氣相色譜儀 原子熒光光譜儀 可見分光光度計 液質聯(lián)用儀 壓力試驗機 酸度計（PH計） 離心機 高速離心機 冷凍離心機 生物顯微鏡 金相顯微鏡 標準物質 生物試劑